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Swiss Institute of Bioinformatics
SwissTargetPrediction
Query Molecule






Target Classes
Top 15
Top 25
Top 50
All
Export results:
Target | Common name | Uniprot ID | ChEMBL ID | Target Class | Probability* | Known actives (3D/2D) |
---|---|---|---|---|---|---|
Neuronal acetylcholine receptor protein alpha-7 subunit | CHRNA7 | P36544 | CHEMBL2492 | Ligand-gated ion channel | 0.147106563998 |
207 /
14   |
Dopamine transporter | SLC6A3 | Q01959 | CHEMBL238 | Electrochemical transporter | 0.112450964818 |
1629 /
495   |
Norepinephrine transporter | SLC6A2 | P23975 | CHEMBL222 | Electrochemical transporter | 0.103761755413 |
949 /
59   |
Serotonin transporter | SLC6A4 | P31645 | CHEMBL228 | Electrochemical transporter | 0.103761755413 |
1785 /
319   |
Butyrylcholinesterase | BCHE | P06276 | CHEMBL1914 | Hydrolase | 0.0864426933852 |
26 /
11   |
Neuronal acetylcholine receptor; alpha4/beta2 | CHRNA4 CHRNB2 | P43681 P17787 | CHEMBL1907589 | Ligand-gated ion channel | 0.0690974435253 |
254 /
12   |
Muscarinic acetylcholine receptor M4 | CHRM4 | P08173 | CHEMBL1821 | Family A G protein-coupled receptor | 0.0690974435253 |
138 /
25   |
Muscarinic acetylcholine receptor M2 | CHRM2 | P08172 | CHEMBL211 | Family A G protein-coupled receptor | 0.0690974435253 |
324 /
62   |
Muscarinic acetylcholine receptor M1 | CHRM1 | P11229 | CHEMBL216 | Family A G protein-coupled receptor | 0.0690974435253 |
468 /
149   |
Muscarinic acetylcholine receptor M3 | CHRM3 | P20309 | CHEMBL245 | Family A G protein-coupled receptor | 0.0690974435253 |
267 /
54   |
Serotonin 3a (5-HT3a) receptor | HTR3A | P46098 | CHEMBL1899 | Ligand-gated ion channel | 0.0690974435253 |
157 /
8   |
Dopamine D3 receptor | DRD3 | P35462 | CHEMBL234 | Family A G protein-coupled receptor | 0.0690974435253 |
365 /
44   |
Serotonin 1b (5-HT1b) receptor (by homology) | HTR1B | P28222 | CHEMBL1898 | Family A G protein-coupled receptor | 0.0604245879294 |
195 /
3   |
Dopamine D2 receptor | DRD2 | P14416 | CHEMBL217 | Family A G protein-coupled receptor | 0.0604245879294 |
1135 /
77   |
Histamine H4 receptor | HRH4 | Q9H3N8 | CHEMBL3759 | Family A G protein-coupled receptor | 0.0604245879294 |
345 /
0   |
Sigma opioid receptor | SIGMAR1 | Q99720 | CHEMBL287 | Membrane receptor | 0.0604245879294 |
621 /
109   |
Serotonin 2c (5-HT2c) receptor | HTR2C | P28335 | CHEMBL225 | Family A G protein-coupled receptor | 0.0604245879294 |
367 /
6   |
HERG | KCNH2 | Q12809 | CHEMBL240 | Voltage-gated ion channel | 0.0604245879294 |
333 /
21   |
Muscarinic acetylcholine receptor M5 | CHRM5 | P08912 | CHEMBL2035 | Family A G protein-coupled receptor | 0.0604245879294 |
149 /
22   |
Serotonin 1a (5-HT1a) receptor | HTR1A | P08908 | CHEMBL214 | Family A G protein-coupled receptor | 0.0604245879294 |
423 /
12   |
Serotonin 2a (5-HT2a) receptor | HTR2A | P28223 | CHEMBL224 | Family A G protein-coupled receptor | 0.0604245879294 |
611 /
12   |
Serotonin 2b (5-HT2b) receptor | HTR2B | P41595 | CHEMBL1833 | Family A G protein-coupled receptor | 0.0604245879294 |
159 /
5   |
Acetylcholinesterase | ACHE | P22303 | CHEMBL220 | Hydrolase | 0.0604245879294 |
116 /
13   |
Mu opioid receptor | OPRM1 | P35372 | CHEMBL233 | Family A G protein-coupled receptor | 0.0604245879294 |
372 /
44   |
Alpha-2a adrenergic receptor | ADRA2A | P08913 | CHEMBL1867 | Family A G protein-coupled receptor | 0.0604245879294 |
41 /
6   |
Alpha-2b adrenergic receptor | ADRA2B | P18089 | CHEMBL1942 | Family A G protein-coupled receptor | 0.0604245879294 |
26 /
6   |
Dopamine D4 receptor | DRD4 | P21917 | CHEMBL219 | Family A G protein-coupled receptor | 0.0604245879294 |
266 /
37   |
Histamine H1 receptor | HRH1 | P35367 | CHEMBL231 | Family A G protein-coupled receptor | 0.0604245879294 |
189 /
12   |
Serotonin 6 (5-HT6) receptor | HTR6 | P50406 | CHEMBL3371 | Family A G protein-coupled receptor | 0.0604245879294 |
279 /
4   |
Adrenergic receptor alpha-2 | ADRA2C | P18825 | CHEMBL1916 | Family A G protein-coupled receptor | 0.0604245879294 |
49 /
5   |
Histamine H2 receptor | HRH2 | P25021 | CHEMBL1941 | Family A G protein-coupled receptor | 0.0604245879294 |
22 /
4   |
Dopamine D1 receptor | DRD1 | P21728 | CHEMBL2056 | Family A G protein-coupled receptor | 0.0604245879294 |
149 /
3   |
Alpha-1d adrenergic receptor | ADRA1D | P25100 | CHEMBL223 | Family A G protein-coupled receptor | 0.0604245879294 |
47 /
6   |
Alpha-1a adrenergic receptor (by homology) | ADRA1A | P35348 | CHEMBL229 | Family A G protein-coupled receptor | 0.0604245879294 |
124 /
7   |
Adenosine A3 receptor | ADORA3 | P0DMS8 | CHEMBL256 | Family A G protein-coupled receptor | 0.0604245879294 |
61 /
3   |
Calcium-activated potassium channel subunit alpha-1 | KCNMA1 | Q12791 | CHEMBL4304 | Voltage-gated ion channel | 0.0604245879294 |
1 /
0   |
C-C motif chemokine 2 | CCL2 | P13500 | CHEMBL1649052 | Family A G protein-coupled receptor | 0.0604245879294 |
3 /
0   |
Neuronal acetylcholine receptor; alpha3/beta4 | CHRNA3 CHRNB4 | P32297 P30926 | CHEMBL1907594 | Ligand-gated ion channel | 0.0604245879294 |
120 /
0   |
Rho-associated protein kinase | ROCK2 ROCK1 | O75116 Q13464 | CHEMBL2111459 | Kinase | 0.0604245879294 |
51 /
0   |
Myosin light chain kinase, smooth muscle | MYLK | Q15746 | CHEMBL2428 | Kinase | 0.0604245879294 |
3 /
0   |
Rho-associated protein kinase 2 | ROCK2 | O75116 | CHEMBL2973 | Kinase | 0.0604245879294 |
128 /
0   |
Protein kinase N2 | PKN2 | Q16513 | CHEMBL3032 | Kinase | 0.0604245879294 |
7 /
0   |
Bromodomain adjacent to zinc finger domain protein 2A | BAZ2A | Q9UIF9 | CHEMBL3108642 | Reader | 0.0604245879294 |
8 /
0   |
Rho-associated protein kinase 1 | ROCK1 | Q13464 | CHEMBL3231 | Kinase | 0.0604245879294 |
45 /
0   |
Protein kinase N1 | PKN1 | Q16512 | CHEMBL3384 | Kinase | 0.0604245879294 |
5 /
0   |
Ribosomal protein S6 kinase alpha 5 | RPS6KA5 | O75582 | CHEMBL4237 | Kinase | 0.0604245879294 |
4 /
0   |
Epidermal growth factor receptor erbB1 | EGFR | P00533 | CHEMBL203 | Kinase | 0.0604245879294 |
123 /
4   |
Neuronal acetylcholine receptor; alpha3/beta2 | CHRNA3 CHRNB2 | P32297 P17787 | CHEMBL2109234 | Ligand-gated ion channel | 0.0604245879294 |
10 /
0   |
Neuronal acetylcholine receptor; alpha3/alpha6/beta2/beta3 | CHRNB3 CHRNA6 CHRNB2 CHRNA3 | Q05901 Q15825 P17787 P32297 | CHEMBL2109233 | Ligand-gated ion channel | 0.0604245879294 |
7 /
0   |
Fibroblast activation protein alpha | FAP | Q12884 | CHEMBL4683 | Protease | 0.0604245879294 |
39 /
0   |
Serotonin 1f (5-HT1f) receptor | HTR1F | P30939 | CHEMBL1805 | Family A G protein-coupled receptor | 0.0604245879294 |
61 /
0   |
Serine/threonine-protein kinase AKT | AKT1 | P31749 | CHEMBL4282 | Kinase | 0.0604245879294 |
46 /
0   |
Monoamine oxidase B | MAOB | P27338 | CHEMBL2039 | Oxidoreductase | 0.0604245879294 |
41 /
0   |
Histamine H3 receptor | HRH3 | Q9Y5N1 | CHEMBL264 | Family A G protein-coupled receptor | 0.0604245879294 |
363 /
57   |
Huntingtin | HTT | P42858 | CHEMBL5514 | Unclassified protein | 0.0604245879294 |
9 /
0   |
Poly [ADP-ribose] polymerase-1 | PARP1 | P09874 | CHEMBL3105 | Enzyme | 0.0604245879294 |
242 /
0   |
Nitric oxide synthase, inducible | NOS2 | P35228 | CHEMBL4481 | Enzyme | 0.0604245879294 |
67 /
0   |
Myeloperoxidase | MPO | P05164 | CHEMBL2439 | Enzyme | 0.0604245879294 |
6 /
0   |
Tyrosine-protein kinase JAK1 | JAK1 | P23458 | CHEMBL2835 | Kinase | 0.0604245879294 |
74 /
0   |
Tyrosine-protein kinase JAK2 | JAK2 | O60674 | CHEMBL2971 | Kinase | 0.0604245879294 |
61 /
0   |
Quinone reductase 2 | NQO2 | P16083 | CHEMBL3959 | Enzyme | 0.0604245879294 |
26 /
0   |
Phosphodiesterase 8B | PDE8B | O95263 | CHEMBL4408 | Phosphodiesterase | 0.0604245879294 |
3 /
0   |
Leukocyte elastase | ELANE | P08246 | CHEMBL248 | Protease | 0.0604245879294 |
13 /
0   |
Melanocortin receptor 4 | MC4R | P32245 | CHEMBL259 | Family A G protein-coupled receptor | 0.0604245879294 |
16 /
0   |
Beta-3 adrenergic receptor | ADRB3 | P13945 | CHEMBL246 | Family A G protein-coupled receptor | 0.0604245879294 |
2 /
1   |
Nitric-oxide synthase, brain | NOS1 | P29475 | CHEMBL3568 | Enzyme | 0.0604245879294 |
88 /
0   |
Serotonin 5a (5-HT5a) receptor (by homology) | HTR5A | P47898 | CHEMBL3426 | Family A G protein-coupled receptor | 0.0604245879294 |
24 /
0   |
Amine oxidase, copper containing | AOC3 | Q16853 | CHEMBL3437 | Enzyme | 0.0604245879294 |
9 /
0   |
Protein kinase C theta | PRKCQ | Q04759 | CHEMBL3920 | Kinase | 0.0604245879294 |
74 /
0   |
Leukocyte proteinase 3 (by homology) | PRTN3 | P24158 | CHEMBL3900 | Protease | 0.0604245879294 |
1 /
0   |
Leucine-rich repeat serine/threonine-protein kinase 2 | LRRK2 | Q5S007 | CHEMBL1075104 | Kinase | 0.0604245879294 |
6 /
0   |
Interleukin-1 receptor-associated kinase 4 | IRAK4 | Q9NWZ3 | CHEMBL3778 | Kinase | 0.0604245879294 |
48 /
0   |
Tyrosine-protein kinase JAK3 | JAK3 | P52333 | CHEMBL2148 | Kinase | 0.0604245879294 |
33 /
0   |
Tyrosine-protein kinase TYK2 | TYK2 | P29597 | CHEMBL3553 | Kinase | 0.0604245879294 |
17 /
0   |
Quinone reductase 1 | NQO1 | P15559 | CHEMBL3623 | Enzyme | 0.0604245879294 |
5 /
0   |
Poly [ADP-ribose] polymerase 2 | PARP2 | Q9UGN5 | CHEMBL5366 | Enzyme | 0.0604245879294 |
29 /
0   |
Solute carrier family 22 member 2 | SLC22A2 | O15244 | CHEMBL1743122 | Electrochemical transporter | 0.0604245879294 |
1 /
0   |
Multidrug and toxin extrusion protein 1 | SLC47A1 | Q96FL8 | CHEMBL1743126 | Electrochemical transporter | 0.0604245879294 |
2 /
0   |
Serotonin 3 (5-HT3) receptor | HTR3B HTR3A | O95264 P46098 | CHEMBL2111332 | Ligand-gated ion channel | 0.0604245879294 |
1 /
0   |
Serine/threonine-protein kinase Chk1 | CHEK1 | O14757 | CHEMBL4630 | Kinase | 0.0604245879294 |
99 /
0   |
Sodium channel protein type IV alpha subunit | SCN4A | P35499 | CHEMBL2072 | Voltage-gated ion channel | 0.0 |
11 /
0   |
Inhibitor of nuclear factor kappa B kinase beta subunit | IKBKB | O14920 | CHEMBL1991 | Kinase | 0.0 |
33 /
0   |
Telomerase reverse transcriptase | TERT | O14746 | CHEMBL2916 | Enzyme | 0.0 |
13 /
0   |
Serine/threonine-protein kinase PIM1 | PIM1 | P11309 | CHEMBL2147 | Kinase | 0.0 |
138 /
0   |
Serine/threonine-protein kinase PIM2 | PIM2 | Q9P1W9 | CHEMBL4523 | Kinase | 0.0 |
101 /
0   |
Nicotinic acetylcholine receptor alpha4/beta2/alpha5 | CHRNA5 CHRNB2 CHRNA4 | P30532 P17787 P43681 | CHEMBL3038461 | Ligand-gated ion channel | 0.0 |
1 /
1   |
Bradykinin B2 receptor | BDKRB2 | P30411 | CHEMBL3157 | Family A G protein-coupled receptor | 0.0 |
6 /
0   |
Nitric-oxide synthase, endothelial | NOS3 | P29474 | CHEMBL4803 | Enzyme | 0.0 |
36 /
0   |
Focal adhesion kinase 1 | PTK2 | Q05397 | CHEMBL2695 | Kinase | 0.0 |
2 /
0   |
Serine/threonine-protein kinase PRKX | PRKX | P51817 | CHEMBL5818 | Kinase | 0.0 |
2 /
0   |
PDZ-binding kinase | PBK | Q96KB5 | CHEMBL4896 | Kinase | 0.0 |
22 /
0   |
Urotensin II receptor | UTS2R | Q9UKP6 | CHEMBL3764 | Family A G protein-coupled receptor | 0.0 |
54 /
17   |
Hormone sensitive lipase | LIPE | Q05469 | CHEMBL3590 | Enzyme | 0.0 |
1 /
0   |
Bromodomain-containing protein 4 | BRD4 | O60885 | CHEMBL1163125 | Reader | 0.0 |
19 /
0   |
Histone acetyltransferase PCAF | KAT2B | Q92831 | CHEMBL5500 | Writer | 0.0 |
3 /
0   |
C-C chemokine receptor type 4 | CCR4 | P51679 | CHEMBL2414 | Family A G protein-coupled receptor | 0.0 |
8 /
0   |
Protein kinase C iota | PRKCI | P41743 | CHEMBL2598 | Kinase | 0.0 |
52 /
0   |
Inhibitor of NF-kappa-B kinase (IKK) | CHUK | O15111 | CHEMBL3476 | Kinase | 0.0 |
11 /
0   |
Kappa Opioid receptor | OPRK1 | P41145 | CHEMBL237 | Family A G protein-coupled receptor | 0.0 |
319 /
22   |
Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET | RET | P07949 | CHEMBL2041 | Kinase | 0.0 |
15 /
0   |
*Probability for the query molecule - assumed as bioactive - to have this protein as target.