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Swiss Institute of Bioinformatics
SwissTargetPrediction
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Query Molecule
Target Classes
Top 15
Top 25
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Export results:
Target | Common name | Uniprot ID | ChEMBL ID | Target Class | Probability* | Known actives (3D/2D) |
---|---|---|---|---|---|---|
Serotonin transporter | SLC6A4 | P31645 | CHEMBL228 | Electrochemical transporter | 1.0 |
1486 /
862   |
Sigma opioid receptor | SIGMAR1 | Q99720 | CHEMBL287 | Membrane receptor | 1.0 |
627 /
717   |
Dopamine D2 receptor (by homology) | DRD2 | P14416 | CHEMBL217 | Family A G protein-coupled receptor | 0.673980204067 |
1102 /
1097   |
Neuronal acetylcholine receptor; alpha4/beta2 | CHRNA4 CHRNB2 | P43681 P17787 | CHEMBL1907589 | Ligand-gated ion channel | 0.428280861155 |
178 /
38   |
Neuronal acetylcholine receptor; alpha3/beta4 | CHRNA3 CHRNB4 | P32297 P30926 | CHEMBL1907594 | Ligand-gated ion channel | 0.428280861155 |
96 /
19   |
Neuronal acetylcholine receptor protein alpha-7 subunit | CHRNA7 | P36544 | CHEMBL2492 | Ligand-gated ion channel | 0.428280861155 |
131 /
8   |
Mu opioid receptor | OPRM1 | P35372 | CHEMBL233 | Family A G protein-coupled receptor | 0.362674718576 |
672 /
1730   |
Dopamine D4 receptor | DRD4 | P21917 | CHEMBL219 | Family A G protein-coupled receptor | 0.329868485421 |
224 /
127   |
Dopamine D3 receptor | DRD3 | P35462 | CHEMBL234 | Family A G protein-coupled receptor | 0.329868485421 |
410 /
543   |
Serotonin 1a (5-HT1a) receptor | HTR1A | P08908 | CHEMBL214 | Family A G protein-coupled receptor | 0.321690506669 |
445 /
249   |
Kappa Opioid receptor | OPRK1 | P41145 | CHEMBL237 | Family A G protein-coupled receptor | 0.313572766871 |
483 /
1035   |
Delta opioid receptor | OPRD1 | P41143 | CHEMBL236 | Family A G protein-coupled receptor | 0.288928252457 |
481 /
1407   |
Glutamate NMDA receptor; GRIN1/GRIN2A | GRIN2A GRIN1 | Q12879 Q05586 | CHEMBL1907604 | Ligand-gated ion channel | 0.280808559877 |
5 /
10   |
Norepinephrine transporter | SLC6A2 | P23975 | CHEMBL222 | Electrochemical transporter | 0.239574695827 |
932 /
423   |
Dopamine transporter | SLC6A3 | Q01959 | CHEMBL238 | Electrochemical transporter | 0.239574695827 |
1299 /
774   |
Dopamine D1 receptor | DRD1 | P21728 | CHEMBL2056 | Family A G protein-coupled receptor | 0.215238178243 |
175 /
184   |
Alpha-1d adrenergic receptor | ADRA1D | P25100 | CHEMBL223 | Family A G protein-coupled receptor | 0.157929217109 |
13 /
35   |
Alpha-1a adrenergic receptor | ADRA1A | P35348 | CHEMBL229 | Family A G protein-coupled receptor | 0.157929217109 |
22 /
82   |
Alpha-1b adrenergic receptor | ADRA1B | P35368 | CHEMBL232 | Family A G protein-coupled receptor | 0.141522086267 |
15 /
55   |
Serotonin 5a (5-HT5a) receptor | HTR5A | P47898 | CHEMBL3426 | Family A G protein-coupled receptor | 0.133337961498 |
33 /
23   |
Dopamine D5 receptor | DRD5 | P21918 | CHEMBL1850 | Family A G protein-coupled receptor | 0.133337961498 |
75 /
67   |
Muscarinic acetylcholine receptor M2 | CHRM2 | P08172 | CHEMBL211 | Family A G protein-coupled receptor | 0.133337961498 |
153 /
57   |
11-beta-hydroxysteroid dehydrogenase 1 | HSD11B1 | P28845 | CHEMBL4235 | Enzyme | 0.125142648574 |
26 /
286   |
Anti-estrogen binding site (AEBS) | EBP | Q15125 | CHEMBL4931 | Enzyme | 0.125142648574 |
3 /
13   |
Muscarinic acetylcholine receptor M1 | CHRM1 | P11229 | CHEMBL216 | Family A G protein-coupled receptor | 0.116965063224 |
257 /
47   |
Synaptic vesicular amine transporter (by homology) | SLC18A2 | Q05940 | CHEMBL1893 | Electrochemical transporter | 0.116965063224 |
17 /
162   |
Serotonin 1b (5-HT1b) receptor (by homology) | HTR1B | P28222 | CHEMBL1898 | Family A G protein-coupled receptor | 0.108770969359 |
169 /
52   |
Steroid 5-alpha-reductase 1 | SRD5A1 | P18405 | CHEMBL1787 | Oxidoreductase | 0.108770969359 |
0 /
33   |
Glutamate [NMDA] receptor subunit epsilon 2 | GRIN2B | Q13224 | CHEMBL1904 | Ligand-gated ion channel | 0.108770969359 |
8 /
18   |
Serotonin 2c (5-HT2c) receptor | HTR2C | P28335 | CHEMBL225 | Family A G protein-coupled receptor | 0.108770969359 |
242 /
133   |
Serotonin 2a (5-HT2a) receptor | HTR2A | P28223 | CHEMBL224 | Family A G protein-coupled receptor | 0.100578902067 |
490 /
387   |
Alpha-2a adrenergic receptor | ADRA2A | P08913 | CHEMBL1867 | Family A G protein-coupled receptor | 0.100578902067 |
16 /
18   |
Adrenergic receptor alpha-2 | ADRA2C | P18825 | CHEMBL1916 | Family A G protein-coupled receptor | 0.100578902067 |
30 /
23   |
Serotonin 2b (5-HT2b) receptor | HTR2B | P41595 | CHEMBL1833 | Family A G protein-coupled receptor | 0.100578902067 |
128 /
86   |
Histamine H2 receptor | HRH2 | P25021 | CHEMBL1941 | Family A G protein-coupled receptor | 0.100578902067 |
17 /
21   |
Serotonin 7 (5-HT7) receptor | HTR7 | P34969 | CHEMBL3155 | Family A G protein-coupled receptor | 0.100578902067 |
170 /
35   |
Dipeptidyl peptidase IV | DPP4 | P27487 | CHEMBL284 | Protease | 0.100578902067 |
461 /
103   |
DNA polymerase alpha subunit | POLA1 | P09884 | CHEMBL1828 | Transferase | 0.100578902067 |
1 /
13   |
Alpha-2b adrenergic receptor | ADRA2B | P18089 | CHEMBL1942 | Family A G protein-coupled receptor | 0.100578902067 |
16 /
15   |
Histamine H3 receptor | HRH3 | Q9Y5N1 | CHEMBL264 | Family A G protein-coupled receptor | 0.100578902067 |
248 /
296   |
Serotonin 1d (5-HT1d) receptor | HTR1D | P28221 | CHEMBL1983 | Family A G protein-coupled receptor | 0.100578902067 |
127 /
48   |
Lysine-specific histone demethylase 1 | KDM1A | O60341 | CHEMBL6136 | Eraser | 0.100578902067 |
73 /
55   |
Adenosine A3 receptor | ADORA3 | P0DMS8 | CHEMBL256 | Family A G protein-coupled receptor | 0.100578902067 |
3 /
5   |
Neuropeptide Y receptor type 5 | NPY5R | Q15761 | CHEMBL4561 | Family A G protein-coupled receptor | 0.100578902067 |
2 /
40   |
Voltage-gated L-type calcium channel alpha-1C subunit | CACNA1C | Q13936 | CHEMBL1940 | Voltage-gated ion channel | 0.100578902067 |
0 /
3   |
P-glycoprotein 1 | ABCB1 | P08183 | CHEMBL4302 | Primary active transporter | 0.100578902067 |
5 /
52   |
HERG | KCNH2 | Q12809 | CHEMBL240 | Voltage-gated ion channel | 0.100578902067 |
239 /
118   |
Acetylcholinesterase | ACHE | P22303 | CHEMBL220 | Hydrolase | 0.100578902067 |
75 /
210   |
Melatonin receptor 1A | MTNR1A | P48039 | CHEMBL1945 | Family A G protein-coupled receptor | 0.100578902067 |
2 /
167   |
Melatonin receptor 1B | MTNR1B | P49286 | CHEMBL1946 | Family A G protein-coupled receptor | 0.100578902067 |
4 /
155   |
Putative hydrolase RBBP9 | RBBP9 | O75884 | CHEMBL1075121 | Enzyme | 0.100578902067 |
0 /
1   |
Small conductance calcium-activated potassium channel protein 1 | KCNN1 | Q92952 | CHEMBL2369 | Voltage-gated ion channel | 0.100578902067 |
0 /
1   |
Small conductance calcium-activated potassium channel protein 3 | KCNN3 | Q9UGI6 | CHEMBL3381 | Voltage-gated ion channel | 0.100578902067 |
0 /
1   |
Small conductance calcium-activated potassium channel protein 2 | KCNN2 | Q9H2S1 | CHEMBL4469 | Voltage-gated ion channel | 0.100578902067 |
0 /
1   |
Toll-like receptor 4 (by homology) | TLR4 | O00206 | CHEMBL5255 | Toll-like and Il-1 receptors | 0.100578902067 |
0 /
11   |
Histamine H1 receptor | HRH1 | P35367 | CHEMBL231 | Family A G protein-coupled receptor | 0.100578902067 |
130 /
45   |
Solute carrier family 22 member 1 | SLC22A1 | O15245 | CHEMBL5685 | Electrochemical transporter | 0.100578902067 |
0 /
1   |
Nociceptin receptor | OPRL1 | P41146 | CHEMBL2014 | Family A G protein-coupled receptor | 0.100578902067 |
181 /
93   |
PH domain leucine-rich repeat-containing protein phosphatase 2 | PHLPP2 | Q6ZVD8 | CHEMBL1275209 | Enzyme | 0.100578902067 |
1 /
0   |
LXR-alpha | NR1H3 | Q13133 | CHEMBL2808 | Nuclear receptor | 0.100578902067 |
0 /
25   |
LXR-beta | NR1H2 | P55055 | CHEMBL4093 | Nuclear receptor | 0.100578902067 |
0 /
24   |
Sodium channel protein type IV alpha subunit | SCN4A | P35499 | CHEMBL2072 | Voltage-gated ion channel | 0.100578902067 |
13 /
0   |
Rho-associated protein kinase 1 | ROCK1 | Q13464 | CHEMBL3231 | Kinase | 0.100578902067 |
27 /
0   |
Rho-associated protein kinase 2 | ROCK2 | O75116 | CHEMBL2973 | Kinase | 0.100578902067 |
93 /
0   |
Neuronal acetylcholine receptor; alpha3/alpha6/beta2/beta3 | CHRNB3 CHRNA6 CHRNB2 CHRNA3 | Q05901 Q15825 P17787 P32297 | CHEMBL2109233 | Ligand-gated ion channel | 0.100578902067 |
7 /
0   |
Serotonin 1e (5-HT1e) receptor | HTR1E | P28566 | CHEMBL2182 | Family A G protein-coupled receptor | 0.100578902067 |
9 /
0   |
Rho-associated protein kinase | ROCK2 ROCK1 | O75116 Q13464 | CHEMBL2111459 | Kinase | 0.100578902067 |
50 /
0   |
Muscarinic acetylcholine receptor M5 | CHRM5 | P08912 | CHEMBL2035 | Family A G protein-coupled receptor | 0.100578902067 |
64 /
28   |
Muscarinic acetylcholine receptor M3 | CHRM3 | P20309 | CHEMBL245 | Family A G protein-coupled receptor | 0.100578902067 |
104 /
50   |
Tyrosine-protein kinase JAK3 | JAK3 | P52333 | CHEMBL2148 | Kinase | 0.100578902067 |
14 /
0   |
Tyrosine-protein kinase JAK1 | JAK1 | P23458 | CHEMBL2835 | Kinase | 0.100578902067 |
43 /
0   |
Tyrosine-protein kinase JAK2 | JAK2 | O60674 | CHEMBL2971 | Kinase | 0.100578902067 |
33 /
0   |
Tyrosine-protein kinase TYK2 | TYK2 | P29597 | CHEMBL3553 | Kinase | 0.100578902067 |
11 /
0   |
Tyrosine-protein kinase LCK | LCK | P06239 | CHEMBL258 | Kinase | 0.100578902067 |
1 /
1   |
Carbonic anhydrase II | CA2 | P00918 | CHEMBL205 | Lyase | 0.100578902067 |
21 /
24   |
Carbonic anhydrase I | CA1 | P00915 | CHEMBL261 | Lyase | 0.100578902067 |
12 /
17   |
Quinone reductase 2 | NQO2 | P16083 | CHEMBL3959 | Enzyme | 0.100578902067 |
5 /
31   |
Glutamate NMDA receptor; GRIN1/GRIN2B | GRIN1 GRIN2B | Q05586 Q13224 | CHEMBL1907603 | Ligand-gated ion channel | 0.100578902067 |
3 /
22   |
Arachidonate 5-lipoxygenase | ALOX5 | P09917 | CHEMBL215 | Oxidoreductase | 0.100578902067 |
0 /
16   |
Butyrylcholinesterase | BCHE | P06276 | CHEMBL1914 | Hydrolase | 0.100578902067 |
24 /
34   |
Rho GDP-dissociation inhibitor 1 | ARHGDIA | P52565 | CHEMBL3638327 | Unclassified protein | 0.100578902067 |
3 /
0   |
Histamine H4 receptor | HRH4 | Q9H3N8 | CHEMBL3759 | Family A G protein-coupled receptor | 0.100578902067 |
86 /
0   |
Tyrosine-protein kinase FYN | FYN | P06241 | CHEMBL1841 | Kinase | 0.100578902067 |
0 /
2   |
Carbonic anhydrase VII | CA7 | P43166 | CHEMBL2326 | Lyase | 0.100578902067 |
0 /
1   |
Carbonic anhydrase III | CA3 | P07451 | CHEMBL2885 | Lyase | 0.100578902067 |
0 /
1   |
Carbonic anhydrase VI | CA6 | P23280 | CHEMBL3025 | Lyase | 0.100578902067 |
0 /
8   |
Carbonic anhydrase IV | CA4 | P22748 | CHEMBL3729 | Lyase | 0.100578902067 |
0 /
8   |
Carbonic anhydrase XIII | CA13 | Q8N1Q1 | CHEMBL3912 | Lyase | 0.100578902067 |
0 /
1   |
Carbonic anhydrase VB | CA5B | Q9Y2D0 | CHEMBL3969 | Lyase | 0.100578902067 |
0 /
1   |
Carbonic anhydrase VA | CA5A | P35218 | CHEMBL4789 | Lyase | 0.100578902067 |
0 /
1   |
Serotonin 3a (5-HT3a) receptor | HTR3A | P46098 | CHEMBL1899 | Ligand-gated ion channel | 0.100578902067 |
73 /
0   |
Calcium-activated potassium channel subunit alpha-1 | KCNMA1 | Q12791 | CHEMBL4304 | Voltage-gated ion channel | 0.100578902067 |
1 /
0   |
Nitric-oxide synthase, brain | NOS1 | P29475 | CHEMBL3568 | Enzyme | 0.100578902067 |
74 /
0   |
Cytochrome P450 24A1 (by homology) | CYP24A1 | Q07973 | CHEMBL4521 | Enzyme | 0.100578902067 |
0 /
7   |
Indoleamine 2,3-dioxygenase | IDO1 | P14902 | CHEMBL4685 | Enzyme | 0.0 |
1 /
0   |
Serotonin 6 (5-HT6) receptor | HTR6 | P50406 | CHEMBL3371 | Family A G protein-coupled receptor | 0.0 |
214 /
27   |
Neuronal acetylcholine receptor protein alpha-4 subunit | CHRNA4 | P43681 | CHEMBL1882 | Ligand-gated ion channel | 0.0 |
28 /
0   |
Protein tyrosine phosphatase receptor type C-associated protein | PTPRCAP | Q14761 | CHEMBL4806 | Enzyme | 0.0 |
1 /
0   |
Epoxide hydratase | EPHX2 | P34913 | CHEMBL2409 | Protease | 0.0 |
6 /
33   |
Neurokinin 1 receptor | TACR1 | P25103 | CHEMBL249 | Family A G protein-coupled receptor | 0.0 |
62 /
146   |
*Probability for the query molecule - assumed as bioactive - to have this protein as target.